Sunday 
 
 
2:00 pm - 9:00 pm 
	
Arrival and Check-in
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 7:40 pm 
	
Introductory Comments by GRC Staff / Welcome and Introduction from the Chairs
 
 
						
7:40 pm - 9:30 pm 
	
Keynote Session: Antibiotic Resistance and the Need for Novel Antibiotic Therapies 
 
 
 
						
7:40 pm - 7:45 pm 
	
Introduction by Discussion Leader
 
 
						
7:45 pm - 8:10 pm 
	
"Multi-Drug Resistant (MDR) Pathogens Are Driving the Need for New Novel Antibacterials" 
 
 
 
						
8:10 pm - 8:15 pm 
	
Discussion
 
 
						
8:15 pm - 8:40 pm 
	
"GARDP: Working Globally to Address the Antimicrobial Resistance Crisis" 
 
 
 
						
8:40 pm - 8:45 pm 
	
Discussion
 
 
						
8:45 pm - 9:10 pm 
	
"How Heteroresistance Changes Our Understanding of Antibiotic Resistance" 
 
 
 
						
9:10 pm - 9:15 pm 
	
Discussion
 
 
						
9:15 pm - 9:30 pm 
	
General Discussion
 
 
						
	Monday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
9:00 am - 12:30 pm 
	
Novel Approaches to Antibiotic Discovery 
 
 
 
						
9:00 am - 9:05 am 
	
Introduction by Discussion Leader
 
 
						
9:05 am - 9:25 am 
	
"Reviving Natural Products Antibiotic Discovery" 
 
 
 
						
9:25 am - 9:35 am 
	
Discussion
 
 
						
9:35 am - 9:55 am 
	
"Generative Artificial Intelligence for Antibiotic Discovery" 
 
 
 
						
9:55 am - 10:05 am 
	
Discussion
 
 
						
10:05 am - 10:25 am 
	
"AI for Antibiotic Discovery" 
 
 
 
						
10:25 am - 10:35 am 
	
Discussion
 
 
						
10:35 am - 11:05 am 
	
Coffee Break
 
 
						
11:05 am - 11:25 am 
	
"Challenges of Antibacterial Discovery" 
 
 
 
						
11:25 am - 11:35 am 
	
Discussion
 
 
						
11:35 am - 11:55 am 
	
"Systems Chemical Biology Approach to Antibiotic Discovery" 
 
 
 
						
11:55 am - 12:05 pm 
	
Discussion
 
 
						
12:05 pm - 12:15 pm 
	
"Enabling Targeted Protein Degradation in Bacteria" 
 
 
 
						
12:15 pm - 12:20 pm 
	
Discussion
 
 
						
12:20 pm - 12:30 pm 
	
General Discussion
 
 
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 9:30 pm 
	
Targeted Based Approaches to Antibacterial Discovery 
 
 
 
						
7:30 pm - 7:35 pm 
	
Introduction by Discussion Leader
 
 
						
7:35 pm - 7:55 pm 
	
"Antibiotics Preorganized for Ribosomal Binding Overcome Antimicrobial Resistance" 
 
 
 
						
7:55 pm - 8:05 pm 
	
Discussion
 
 
						
8:05 pm - 8:25 pm 
	
"Macrocyclic Peptides Disassemble the Periplasmic LPS Transport Bridge: New Approaches to Kill Multidrug-Resistant Gram-Negative Bacteria" 
 
 
 
						
8:25 pm - 8:35 pm 
	
Discussion
 
 
						
8:35 pm - 8:55 pm 
	
"Cracking Nature’s Recipes to Design Lipid-Targeting Antibiotics" 
 
 
 
						
8:55 pm - 9:05 pm 
	
Discussion
 
 
						
9:05 pm - 9:15 pm 
	
"PBP2:MreC: An Ideal Target for New Antibacterial Agents" 
 
 
 
						
9:15 pm - 9:20 pm 
	
Discussion
 
 
						
9:20 pm - 9:30 pm 
	
General Discussion
 
 
						
	Tuesday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
8:30 am - 9:00 am 
	
Group Photo
 
 
						
9:00 am - 12:30 pm 
	
Discovery Pipelines: Hits, Leads and Candidates 
 
 
 
						
9:00 am - 9:05 am 
	
Introduction by Discussion Leader
 
 
						
9:05 am - 9:25 am 
	
"Discovering Mechanistically Novel Antibacterial Leads through Phenotypic Screening" 
 
 
 
						
9:25 am - 9:35 am 
	
Discussion
 
 
						
9:35 am - 9:55 am 
	
"Development of Broad-Spectrum MBL Inhibitors" 
 
 
 
						
9:55 am - 10:05 am 
	
Discussion
 
 
						
10:05 am - 10:25 am 
	
"Engineering Broad Spectrum Novel Ribosome Inhibitors" 
 
 
 
						
10:25 am - 10:35 am 
	
Discussion
 
 
						
10:35 am - 11:05 am 
	
Coffee Break
 
 
						
11:05 am - 11:25 am 
	
"Attracting New Anti-Infective Candidates with Novel Targets Using the MAGNET Discovery Platform" 
 
 
 
						
11:25 am - 11:35 am 
	
Discussion
 
 
						
11:35 am - 11:55 am 
	
"Achilles Heel of the Trojan Horse: Host Directed Therapy Against Mycobacterial Infections" 
 
 
 
						
11:55 am - 12:05 pm 
	
Discussion
 
 
						
12:05 pm - 12:15 pm 
	
"The Guanidino Lipoglycopeptides: Semisynthetic Glycopeptides with Potent in Vitro and in Vivo Antibacterial Activity" 
 
 
 
						
12:15 pm - 12:20 pm 
	
Discussion
 
 
						
12:20 pm - 12:30 pm 
	
General Discussion
 
 
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 9:30 pm 
	
The Bacterial Cell Envelope: Targets and Requirements for Drug Permeation 
 
 
 
						
7:30 pm - 7:35 pm 
	
Introduction by Discussion Leader
 
 
						
7:35 pm - 7:55 pm 
	
"A New Antibiotic Traps Lipopolysaccharide in its Intermembrane Transporter" 
 
 
 
						
7:55 pm - 8:05 pm 
	
Discussion
 
 
						
8:05 pm - 8:25 pm 
	
"How Do Polymyxins Kill Bacteria?" 
 
 
 
						
8:25 pm - 8:35 pm 
	
Discussion
 
 
						
8:35 pm - 8:55 pm 
	
"Measuring the Interactions of Polymyxins with the Gram-Negative Outer Membrane" 
 
 
 
						
8:55 pm - 9:05 pm 
	
Discussion
 
 
						
9:05 pm - 9:15 pm 
	
"Guidelines for Compound Accumulation in Pseudomonas Aeruginosa Enable Antibiotic Development" 
 
 
 
						
9:15 pm - 9:20 pm 
	
Discussion
 
 
						
9:20 pm - 9:30 pm 
	
General Discussion
 
 
						
	Wednesday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
9:00 am - 12:30 pm 
	
Advances in Antibiotic Combination Therapy 
 
 
 
						
9:00 am - 9:05 am 
	
Introduction by Discussion Leader
 
 
						
9:05 am - 9:25 am 
	
"Beta-Lactamases and Skaters: Pairs and Singles" 
 
 
 
						
9:25 am - 9:35 am 
	
Discussion
 
 
						
9:35 am - 9:55 am 
	
"Mechanistic Insights and Therapeutic Strategies for Targeting the Most Synergistic Penicillin-Binding Proteins Across Three Gram-Negative ‘Superbugs’" 
 
 
 
						
9:55 am - 10:05 am 
	
Discussion
 
 
						
10:05 am - 10:25 am 
	
"Discovery of Enmetazobactam" 
 
 
 
						
10:25 am - 10:35 am 
	
Discussion
 
 
						
10:35 am - 11:05 am 
	
Coffee Break
 
 
						
11:05 am - 11:25 am 
	
"Mycobacterium Abscessus: The Promise of Dual ß-Lactams Therapy" 
 
 
 
						
11:25 am - 11:35 am 
	
Discussion
 
 
						
11:35 am - 11:55 am 
	
"How to Give Bacteria Food Poisoning: Antibiotics that Hijack Nutrient Transporters" 
 
 
 
						
11:55 am - 12:05 pm 
	
Discussion
 
 
						
12:05 pm - 12:15 pm 
	
"Applying Concepts on Antibiotic-Induced Bacterial Death to Rationally Combine Drugs for Treatment of Mycobacterium Abscessus Lung Disease" 
 
 
 
						
12:15 pm - 12:20 pm 
	
Discussion
 
 
						
12:20 pm - 12:30 pm 
	
General Discussion
 
 
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 9:30 pm 
	
Unconventional Antibiotics: Phage Therapy and Anti-Infectives 
 
 
 
						
7:30 pm - 7:35 pm 
	
Introduction by Discussion Leader
 
 
						
7:35 pm - 7:55 pm 
	
"Biasing Bacteriophage Behaviours" 
 
 
 
						
7:55 pm - 8:05 pm 
	
Discussion
 
 
						
8:05 pm - 8:25 pm 
	
"Antisense Antibiotics as Precision Therapeutics for Pseudomonas Aeruginosa" 
 
 
 
						
8:25 pm - 8:35 pm 
	
Discussion
 
 
						
8:35 pm - 8:55 pm 
	
"Development of Efflux Pump Inhibitors for Overcoming Antimicrobial Resistance in Enterobacterales Infections" 
 
 
 
						
8:55 pm - 9:05 pm 
	
Discussion
 
 
						
9:05 pm - 9:15 pm 
	
"Chemical Inhibition of Staphylococcus Aureus  Virulence with a Plant-Derived Natural Product" 
 
 
 
						
9:15 pm - 9:20 pm 
	
Discussion
 
 
						
9:20 pm - 9:30 pm 
	
General Discussion
 
 
						
	Thursday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
8:30 am - 9:00 am 
	
Business Meeting 
Nominations for the Next Vice Chair(s); Complete the GRC Evaluation Forms; Election of the Next Vice Chair(s) 
 
 
						
9:00 am - 12:30 pm 
	
Moving the Needle for Difficult-to-Eradicate Infections 
 
 
 
						
9:00 am - 9:05 am 
	
Introduction by Discussion Leader
 
 
						
9:05 am - 9:35 am 
	
"Addressing Antimicrobial Resistance in Clostridioides difficile : Clinical Implications and the Motivation for Novel Treatment Approaches" 
 
 
 
						
9:35 am - 9:45 am 
	
Discussion
 
 
						
9:45 am - 10:05 am 
	
"A Six Decade Wait for a Novel Broad-Spectrum Antibacterial Drug Class: Development of BWC0977" 
 
 
 
						
10:05 am - 10:15 am 
	
Discussion
 
 
						
10:15 am - 10:45 am 
	
Coffee Break
 
 
						
10:45 am - 11:05 am 
	
"Redesign of Rifamycins for the Treatment of Mycobacterium Abscesuss  Lung Disease" 
 
 
 
						
11:05 am - 11:15 am 
	
Discussion
 
 
						
11:15 am - 11:35 am 
	
"Apramycin, a Promising Candidate in the Treatment of Chronic NTM Infections" 
 
 
 
						
11:35 am - 11:45 am 
	
Discussion
 
 
						
11:45 am - 12:05 pm 
	
"Omadacycline as a Potential New Option for NTM Pulmonary Disease Caused by M. Abscessus " 
 
 
 
						
12:05 pm - 12:15 pm 
	
Discussion
 
 
						
12:15 pm - 12:30 pm 
	
General Discussion
 
 
						
12:30 pm - 1:30 pm 
	
Lunch
 
 
						
1:30 pm - 4:00 pm 
	
Free Time
 
 
						
4:00 pm - 6:00 pm 
	
Poster Session 
 
 
						
6:00 pm - 7:00 pm 
	
Dinner
 
 
						
7:30 pm - 9:30 pm 
	
Learning from Failures and Moving to Success in Clinical Trials 
 
 
 
						
7:30 pm - 7:35 pm 
	
Introduction by Discussion Leader
 
 
						
7:35 pm - 7:55 pm 
	
"Experiences and Learnings through Developing a Novel Antibiotic, Zosurabalpin" 
 
 
 
						
7:55 pm - 8:05 pm 
	
Discussion
 
 
						
8:05 pm - 8:25 pm 
	
"Clinical Data on a Phage Trial" 
 
 
 
						
8:25 pm - 8:35 pm 
	
Discussion
 
 
						
8:35 pm - 9:05 pm 
	
"Integrating Global Needs and R&D Activities to Solve the Antibiotic Resistance Crisis" 
 
 
 
						
9:05 pm - 9:15 pm 
	
Discussion
 
 
						
9:15 pm - 9:30 pm 
	
Closing Remarks
 
 
						
	Friday 
 
 
7:30 am - 8:30 am 
	
Breakfast
 
 
						
9:00 am 
	
Departure